Author: Schirmeister, Tanja and Zappala, Maria / Organizational unit: FB 09 Chemie, Pharmazie, Geographie und Geowissenschaften - Universitätsbibliographie Search Results

Start Over Author Schirmeister, Tanja Author Zappala, Maria Organizational unit FB 09 Chemie, Pharmazie, Geographie und Geowissenschaften

1. Drug Combination Studies of the Dipeptide Nitrile CD24 with Curcumin: A New Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense

Autoren:: Di Chio, Carla; Previti, Santo; De Luca, Fabiola; Bogacz, Marta; Zimmer, Collin; Wagner, Annika; Schirmeister, Tanja; Zappala, Maria; Ettari, Roberta
Veröffentlichungsdatum:: 2022
Type:: Journal article

2. Evaluation of curcumin irreversibility

Autoren:: Ettari, Roberta; Previti, Santo; Maiorana, Santina; Allegra, Alessandro; Schirmeister, Tanja; Grasso, Silvana; Zappala, Maria
Veröffentlichungsdatum:: 2020
Type:: Journal article

3. Novel 2H-isoquinolin-3-ones as antiplasmodial falcipain-2 inhibitors

Autoren:: Micale, Nicola; Ettari, Roberta; Schirmeister, Tanja; Evers, Astrid; Gelhaus, Christoph; Leippe, Matthias; Zappala, Maria; Grasso, Silvana
Veröffentlichungsdatum:: 2009
Type:: Journal article

4. Peptidomimetics containing a vinyl ketone warhead as falcipain-2 inhibitors

Autoren:: Ettari, Roberta; Zappala, Maria; Micale, Nicola; Grazioso, Giovanni; Giofre, Salvatore; Schirmeister, Tanja; Grasso, Silvana
Veröffentlichungsdatum:: 2011
Type:: Journal article

5. Identification of noncovalent proteasome inhibitors with high selectivity for chymotrypsin-like activity by a multistep structure based virtual screening

Autoren:: Di Giovanni, Carmen; Ettari, Roberta; Sarno, Serena; Rotondo, Archimede; Bitto, Alessandra; Squadrito, Francesco; Altavilla, Domenica; Schirmeister, Tanja; Novellino, Ettore; Grasso, Silvana; Zappala, Maria; Lavecchia, Antonio
Veröffentlichungsdatum:: 2016
Type:: Journal article

6. Optimization of peptidomimetic boronates bearing a P3 bicyclic scaffold as proteasome inhibitors

Autoren:: Troiano, Valeria; Scarbaci, Kety; Ettari, Roberta; Micale, Nicola; Cerchia, Carmen; Pinto, Andrea; Schirmeister, Tanja; Novellino, Ettore; Grasso, Silvana; Lavecchia, Antonio; Zappala, Maria
Veröffentlichungsdatum:: 2014
Type:: Journal article

7. Identification of a new series of amides as non-covalent proteasome inhibitors

Autoren:: Scarbaci, Kety; Troiano, Valeria; Micale, Nicola; Ettari, Roberta; Tamborini, Lucia; Di Giovanni, Carmen; Cerchia, Carmen; Grasso, Silvana; Novellino, Ettore; Schirmeister, Tanja; Lavecchia, Antonio; Zappala, Maria
Veröffentlichungsdatum:: 2014
Type:: Journal article

8. Development of peptidomimetic boronates as proteasome inhibitors

Autoren:: Micale, Nicola; Ettari, Roberta; Lavecchia, Antonio; Di Giovanni, Carmen; Scarbaci, Kety; Troiano, Valeria; Grasso, Silvana; Novellino, Ettore; Schirmeister, Tanja; Zappala, Maria
Veröffentlichungsdatum:: 2013
Type:: Journal article

9. Drug synergism: studies of combination of RK-52 and curcumin against rhodesain of Trypanosoma brucei rhodesiense

Autoren:: Ettari, Roberta; Previti, Santo; Di Chio, Carla; Maiorana, Santina; Allegra, Alessandro; Schirmeister, Tanja; Zappala, Maria
Veröffentlichungsdatum:: 2020
Type:: Journal article

10. Lead discovery of SARS-CoV-2 main protease inhibitors through covalent docking-based virtual screening

Autoren:: Amendola, Giorgio; Ettari, Roberta; Santo, Previti; Di Chio, Carla; Messere, Anna; Di Maro, Salvatore; Hammerschmidt, Stefan J; Zimmer, Collin; Zimmermann, Robert A; Schirmeister, Tanja; Zappala, Maria; Cosconati, Sandro
Veröffentlichungsdatum:: 2021
Type:: Journal article