Author: Micale, Nicola / Organizational unit: Institut für Pharmazeutische und Biomedizinische Wissenschaften and Pharmazeutische/Medizinische Chemie 1 / Data source: PubMed - Universitätsbibliographie Search Results

Start Over Author Micale, Nicola Organizational unit Institut für Pharmazeutische und Biomedizinische Wissenschaften Organizational unit Pharmazeutische/Medizinische Chemie 1 Data source PubMed

1. Novel 2H-isoquinolin-3-ones as antiplasmodial falcipain-2 inhibitors

Autoren:: Micale, Nicola; Ettari, Roberta; Schirmeister, Tanja; Evers, Astrid; Gelhaus, Christoph; Leippe, Matthias; Zappala, Maria; Grasso, Silvana
Veröffentlichungsdatum:: 2009
Type:: Journal article

2. Gold compounds as cysteine protease inhibitors: perspectives for pharmaceutical application as antiparasitic agents

Autoren:: Massai, Lara; Messori, Luigi; Micale, Nicola; Schirmeister, Tanja; Maes, Louis; Fregona, Dolores; Cinellu, Maria Agostina; Gabbiani, Chiara
Veröffentlichungsdatum:: 2017
Type:: Journal article

3. Selected cytotoxic gold compounds cause significant inhibition of 20S proteasome catalytic activities

Autoren:: Micale, Nicola; Schirmeister, Tanja; Ettari, Roberta; Cinellu, Maria A; Maiore, Laura; Serratrice, Maria; Gabbiani, Chiara; Massai, Lara; Messori, Luigi
Veröffentlichungsdatum:: 2014
Type:: Journal article

4. Selected gold compounds cause pronounced inhibition of Falcipain 2 and effectively block P. falciparum growth in vitro

Autoren:: Micale, Nicola; Cinellu, Maria Agostina; Maiore, Laura; Sannella, Anna Rosa; Severini, Carlo; Schirmeister, Tanja; Gabbiani, Chiara; Messori, Luigi
Veröffentlichungsdatum:: 2011
Type:: Journal article

5. Peptidomimetics containing a vinyl ketone warhead as falcipain-2 inhibitors

Autoren:: Ettari, Roberta; Zappala, Maria; Micale, Nicola; Grazioso, Giovanni; Giofre, Salvatore; Schirmeister, Tanja; Grasso, Silvana
Veröffentlichungsdatum:: 2011
Type:: Journal article

6. Synthesis of C3/C1-Substituted Tetrahydroisoquinolines

Autoren:: Mihoubi, Mohamed; Micale, Nicola; Scala, Angela; Jarraya, Raoudha Mezghani; Bouaziz, Amira; Schirmeister, Tanja; Risitano, Francesco; Piperno, Anna; Grassi, Giovanni
Veröffentlichungsdatum:: 2015
Type:: Journal article

7. Optimization of peptidomimetic boronates bearing a P3 bicyclic scaffold as proteasome inhibitors

Autoren:: Troiano, Valeria; Scarbaci, Kety; Ettari, Roberta; Micale, Nicola; Cerchia, Carmen; Pinto, Andrea; Schirmeister, Tanja; Novellino, Ettore; Grasso, Silvana; Lavecchia, Antonio; Zappala, Maria
Veröffentlichungsdatum:: 2014
Type:: Journal article

8. Identification of a new series of amides as non-covalent proteasome inhibitors

Autoren:: Scarbaci, Kety; Troiano, Valeria; Micale, Nicola; Ettari, Roberta; Tamborini, Lucia; Di Giovanni, Carmen; Cerchia, Carmen; Grasso, Silvana; Novellino, Ettore; Schirmeister, Tanja; Lavecchia, Antonio; Zappala, Maria
Veröffentlichungsdatum:: 2014
Type:: Journal article

9. Development of peptidomimetic boronates as proteasome inhibitors

Autoren:: Micale, Nicola; Ettari, Roberta; Lavecchia, Antonio; Di Giovanni, Carmen; Scarbaci, Kety; Troiano, Valeria; Grasso, Silvana; Novellino, Ettore; Schirmeister, Tanja; Zappala, Maria
Veröffentlichungsdatum:: 2013
Type:: Journal article

10. Nonpeptidic vinyl and allyl phosphonates as falcipain-2 inhibitors

Autoren:: Ettari, Roberta; Nizi, Emanuela; Di Francesco, Maria Emilia; Micale, Nicola; Grasso, Silvana; Zappala, Maria; Vicik, Radim; Schirmeister, Tanja
Veröffentlichungsdatum:: 2008
Type:: Journal article