Author: Kersten, Christian and Schirmeister, Tanja / Organizational unit: FB 09 Chemie, Pharmazie, Geographie und Geowissenschaften / Data source: Europe PubMed Central - Universitätsbibliographie Search Results

Start Over Author Kersten, Christian Author Schirmeister, Tanja Organizational unit FB 09 Chemie, Pharmazie, Geographie und Geowissenschaften Data source Europe PubMed Central

1. Protease detection in the biosensor era: A review

Autoren:: Rai, Pratika; Hoba, Sabrina N; Buchmann, Celine; Subirana-Slotos, Robert J; Kersten, Christian; Schirmeister, Tanja; Endres, Kristina; Bufe, Bernd; Tarasov, Alexey
Veröffentlichungsdatum:: 2024
Type:: Journal article

2. Chemical Space Virtual Screening against Hard-to-Drug RNA Methyltransferases DNMT2 and NSUN6

Autoren:: Zimmermann, Robert A; Fischer, Tim R; Schwickert, Marvin; Nidoieva, Zarina; Schirmeister, Tanja; Kersten, Christian
Veröffentlichungsdatum:: 2023
Type:: Journal article

3. Investigation of the Compatibility between Warheads and Peptidomimetic Sequences of Protease Inhibitors-A Comprehensive Reactivity and Selectivity Study

Autoren:: Mueller, Patrick; Meta, Mergim; Meidner, Jan Laurenz; Schwickert, Marvin; Meyr, Jessica; Schwickert, Kevin; Kersten, Christian; Zimmer, Collin; Hammerschmidt, Stefan Josef; Frey, Ariane; Lahu, Albin; de la Hoz-Rodriguez, Sergio; Agost-Beltran, Laura; Rodriguez, Santiago; Diemer, Kira; Neumann, Wilhelm; Gonzalez, Florenci V; Engels, Bernd; Schirmeister, Tanja
Veröffentlichungsdatum:: 2023
Type:: Journal article

4. Proline-Based Allosteric Inhibitors of Zika and Dengue Virus NS2B/NS3 Proteases

Autoren:: Millies, Benedikt; von Hammerstein, Franziska; Gellert, Andrea; Hammerschmidt, Stefan; Barthels, Fabian; Goeppel, Ulrike; Immerheiser, Melissa; Elgner, Fabian; Jung, Nathalie; Basic, Michael; Kersten, Christian; Kiefer, Werner; Bodem, Jochen; Hildt, Eberhard; Windbergs, Maike; Hellmich, Ute A; Schirmeister, Tanja
Veröffentlichungsdatum:: 2019
Type:: Journal article

5. Warhead Reactivity Limits the Speed of Inhibition of the Cysteine Protease Rhodesain

Autoren:: Johe, Patrick; Jung, Sascha; Endres, Erik; Kersten, Christian; Zimmer, Collin; Ye, Weixiang; Soennichsen, Carsten; Hellmich, Ute A; Sotriffer, Christoph; Schirmeister, Tanja; Neuweiler, Hannes
Veröffentlichungsdatum:: 2021
Type:: Journal article

6. New aziridine-based inhibitors of cathepsin L-like cysteine proteases with selectivity for the Leishmania cysteine protease LmCPB2.8

Autoren:: Fey, Philipp; Chartomatsidou, Roula; Kiefer, Werner; Mottram, Jeremy C; Kersten, Christian; Schirmeister, Tanja
Veröffentlichungsdatum:: 2018
Type:: Journal article

7. Structure, interdomain dynamics, and pH-dependent autoactivation of pro-rhodesain, the main lysosomal cysteine protease from African trypanosomes

Autoren:: Johe, Patrick; Jaenicke, Elmar; Neuweiler, Hannes; Schirmeister, Tanja; Kersten, Christian; Hellmich, Ute A
Veröffentlichungsdatum:: 2021
Type:: Journal article

8. Structure, interdomain dynamics and pH-dependent autoactivation of pro-rhodesain, the main lysosomal cysteine protease from African trypanosomes

Autoren:: Johé, Patrick; Jaenicke, Elmar; Neuweiler, Hannes; Schirmeister, Tanja; Kersten, Christian; Hellmich, Ute A
Veröffentlichungsdatum:: 2020
Type:: Preprint

9. Interface with Host Proteases in SARS-CoV-2 Entry as a Promising Therapeutic Strategy

Autoren:: Mueller, Patrick; Maus, Hannah; Hammerschmidt, Stefan Josef; Knaff, Philip; Mailaender, Volker; Schirmeister, Tanja; Kersten, Christian
Veröffentlichungsdatum:: 2022
Type:: Journal article

10. Fluorovinylsulfones and -Sulfonates as Potent Covalent Reversible Inhibitors of the Trypanosomal Cysteine Protease Rhodesain: Structure-Activity Relationship, Inhibition Mechanism, Metabolism, and In Vivo Studies

Autoren:: Jung, Sascha; Fuchs, Natalie; Johe, Patrick; Wagner, Annika; Diehl, Erika; Yuliani, Tri; Zimmer, Collin; Barthels, Fabian; Zimmermann, Robert A; Klein, Philipp; Waigel, Waldemar; Meyr, Jessica; Opatz, Till; Tenzer, Stefan; Distler, Ute; Raeder, Hans-Joachim; Kersten, Christian; Engels, Bernd; Hellmich, Ute A; Klein, Jochen; Schirmeister, Tanja
Veröffentlichungsdatum:: 2021
Type:: Journal article