Author: 3 selected / Organizational unit: FB 09 Chemie, Pharmazie, Geographie und Geowissenschaften - Universitätsbibliographie Search Results

Start Over Author Cosconati, Sandro Author Schirmeister, Tanja Author Zappala, Maria Organizational unit FB 09 Chemie, Pharmazie, Geographie und Geowissenschaften

1. Development of novel dipeptide nitriles as inhibitors of rhodesain of Trypanosoma brucei rhodesiense

Autoren:: Di Chio, Carla; Previti, Santo; Amendola, Giorgio; Ravichandran, Rahul; Wagner, Annika; Cosconati, Sandro; Hellmich, Ute A; Schirmeister, Tanja; Zappala, Maria; Ettari, Roberta
Veröffentlichungsdatum:: 2022
Type:: Journal article

2. Synthesis and biological evaluation of novel peptidomimetics as rhodesain inhibitors

Autoren:: Ettari, Roberta; Previti, Santo; Cosconati, Sandro; Kesselring, Jochen; Schirmeister, Tanja; Grasso, Silvana; Zappala, Maria
Veröffentlichungsdatum:: 2016
Type:: Journal article

3. Development of novel 1,4-benzodiazepine-based Michael acceptors as antitrypanosomal agents

Autoren:: Ettari, Roberta; Previti, Santo; Cosconati, Sandro; Maiorana, Santina; Schirmeister, Tanja; Grasso, Silvana; Zappala, Maria
Veröffentlichungsdatum:: 2016
Type:: Journal article

4. Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs)

Autoren:: Previti, Santo; Ettari, Roberta; Cosconati, Sandro; Arnendola, Giorgio; Chouchene, Khawla; Wagner, Annika; Hellmich, Ute A; Ulrich, Kathrin; Krauth-Siegel, R Luise; Wich, Peter R; Schmid, Ira; Schirmeister, Tanja; Gut, Jiri; Rosenthal, Philip J; Grasso, Silvana; Zappala, Maria
Veröffentlichungsdatum:: 2017
Type:: Journal article

5. Lead discovery of SARS-CoV-2 main protease inhibitors through covalent docking-based virtual screening

Autoren:: Amendola, Giorgio; Ettari, Roberta; Santo, Previti; Di Chio, Carla; Messere, Anna; Di Maro, Salvatore; Hammerschmidt, Stefan J; Zimmer, Collin; Zimmermann, Robert A; Schirmeister, Tanja; Zappala, Maria; Cosconati, Sandro
Veröffentlichungsdatum:: 2021
Type:: Journal article

6. Development of Novel Benzodiazepine-Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense

Autoren:: Di Chio, Carla; Previti, Santo; Amendola, Giorgio; Cosconati, Sandro; Schirmeister, Tanja; Zappala, Maria; Ettari, Roberta
Veröffentlichungsdatum:: 2020
Type:: Journal article

7. Optimization strategy of novel peptide-based Michael acceptors for the treatment of human African trypanosomiasis

Autoren:: Ettari, Roberta; Previti, Santo; Maiorana, Santina; Amendola, Giorgio; Wagner, Annika; Cosconati, Sandro; Schirmeister, Tanja; Hellmich, Ute A; Zappala, Maria
Veröffentlichungsdatum:: 2019
Type:: Journal article

8. Peptidyl Vinyl Ketone Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment

Autoren:: Maiorana, Santina; Ettari, Roberta; Previti, Santo; Amendola, Giorgio; Wagner, Annika; Cosconati, Sandro; Hellmich, Ute A; Schirmeister, Tanja; Zappala, Maria
Veröffentlichungsdatum:: 2020
Type:: Journal article