work / Autor: Schirmeister, Tanja / Datenquelle: Europe PubMed Central - Universitätsbibliographie Suchergebnisse

Neu anfangen work Autor Schirmeister, Tanja Datenquelle Europe PubMed Central

1. Lead discovery of SARS-CoV-2 main protease inhibitors through covalent docking-based virtual screening

Autoren:: Amendola, Giorgio; Ettari, Roberta; Santo, Previti; Di Chio, Carla; Messere, Anna; Di Maro, Salvatore; Hammerschmidt, Stefan J; Zimmer, Collin; Zimmermann, Robert A; Schirmeister, Tanja; Zappala, Maria; Cosconati, Sandro
Veröffentlichungsdatum:: 2021
Typ:: Zeitschriftenaufsatz

2. The importance of the active site histidine for the activity of epoxide- or aziridine-based inhibitors of cysteine proteases

Autoren:: Mladenovic, Milena; Schirmeister, Tanja; Thiel, Stefan; Thiel, Walter; Engels, Bernd
Veröffentlichungsdatum:: 2007
Typ:: Zeitschriftenaufsatz

3. Synthesis and Biological Evaluation of Papain-Family Cathepsin L-Like Cysteine Protease Inhibitors Containing a 1,4-Benzodiazepine Scaffold as Antiprotozoal Agents

Autoren:: Ettari, Roberta; Pinto, Andrea; Tamborini, Lucia; Angelo, Ilenia C; Grasso, Silvana; Zappala, Maria; Capodicasa, Natale; Yzeiraj, Laura; Gruber, Esther; Aminake, Makoah N; Pradel, Gabriele; Schirmeister, Tanja; De Micheli, Carlo; Conti, Paola
Veröffentlichungsdatum:: 2014
Typ:: Zeitschriftenaufsatz

4. Rational design of aziridine-containing cysteine protease inhibitors with improved potency: Studies on inhibition mechanism

Autoren:: Vicik, Radim; Helten, Holger; Schirmeister, Tanja; Engels, Bernd
Veröffentlichungsdatum:: 2006
Typ:: Zeitschriftenaufsatz

5. Drug Combination Studies of the Dipeptide Nitrile CD24 with Curcumin: A New Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense

Autoren:: Di Chio, Carla; Previti, Santo; De Luca, Fabiola; Bogacz, Marta; Zimmer, Collin; Wagner, Annika; Schirmeister, Tanja; Zappala, Maria; Ettari, Roberta
Veröffentlichungsdatum:: 2022
Typ:: Zeitschriftenaufsatz

6. Effect of Electron-Withdrawing Substituents on the Epoxide Ring: An Experimental and Theoretical Electron Density Analysis of a Series of Epoxide Derivatives

Autoren:: Grabowsky, Simon; Schirmeister, Tanja; Paulmann, Carsten; Pfeuffer, Thomas; Luger, Peter
Veröffentlichungsdatum:: 2011
Typ:: Zeitschriftenaufsatz

7. Identification of a new series of amides as non-covalent proteasome inhibitors

Autoren:: Scarbaci, Kety; Troiano, Valeria; Micale, Nicola; Ettari, Roberta; Tamborini, Lucia; Di Giovanni, Carmen; Cerchia, Carmen; Grasso, Silvana; Novellino, Ettore; Schirmeister, Tanja; Lavecchia, Antonio; Zappala, Maria
Veröffentlichungsdatum:: 2014
Typ:: Zeitschriftenaufsatz

8. On the origin of the stabilization of the zwitterionic resting state of cysteine proteases: A theoretical study

Autoren:: Mladenovic, Milena; Fink, Reinhold F; Thiel, Walter; Schirmeister, Tanja; Engels, Bernd
Veröffentlichungsdatum:: 2008
Typ:: Zeitschriftenaufsatz

9. Impact of the Recognition Part of Dipeptidyl Nitroalkene Compounds on the Inhibition Mechanism of Cysteine Proteases Cruzain and Cathepsin L

Autoren:: Arafet, Kemel; Royo, Santiago; Schirmeister, Tanja; Barthels, Fabian; V. Gonzalez, Florenci; Moliner, Vicent
Veröffentlichungsdatum:: 2023
Typ:: Zeitschriftenaufsatz

10. New aziridine-based inhibitors of cathepsin L-like cysteine proteases with selectivity for the Leishmania cysteine protease LmCPB2.8

Autoren:: Fey, Philipp; Chartomatsidou, Roula; Kiefer, Werner; Mottram, Jeremy C; Kersten, Christian; Schirmeister, Tanja
Veröffentlichungsdatum:: 2018
Typ:: Zeitschriftenaufsatz